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Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition

Simon Hayek , Nicolas Pietrancosta , Anna Hovhannisyan , Rodolphe Alves de Sousa , Nassima Bekaddour , et al.
European Journal of Medicinal Chemistry, 2020, 186, pp.111855. ⟨10.1016/j.ejmech.2019.111855⟩
Journal articles hal-02372490v1
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In silico studies, synthesis and binding evaluation of substituted 2-pyrrolidinones as peptidomimetics of RGD tripeptide sequence

Valérie Toum , Julie Bolley , Yoann Lalatonne , Carole Barbey , Laurence Motte , et al.
European Journal of Medicinal Chemistry, 2015, 93, pp.360. ⟨10.1016/j.ejmech.2015.02.017⟩
Journal articles hal-01904943v1
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Ferrocifens labelled with an infrared rhenium tricarbonyl tag: synthesis, antiproliferative activity, quantification and nano IR mapping in cancer cells

Yong Wang , Franz Heinemann , Siden Top , Alexandre Dazzi , Clotilde Policar , et al.
Dalton Transactions, 2018, 47 (29), pp.9824 - 9833. ⟨10.1039/C8DT01582A⟩
Journal articles hal-01878514v1

Bacterial Transferase MraY, a Source of Inspiration towards New Antibiotics

Mickaël Fer , Laurent Le Corre , Nicolas Pietrancosta , Nathalie Evrard-Todeschi , Samir Olatunji , et al.
Current Medicinal Chemistry, 2018, 25 (42), pp.6013-6029. ⟨10.2174/0929867325666180330095154⟩
Journal articles hal-02364241v1
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Bioorthogonal Conjugation of Transition Organometallic Complexes to Peptides and Proteins: Strategies and Applications

Michèle Salmain , Nathalie Fischer-Durand , Bogna Rudolf
European Journal of Inorganic Chemistry, 2020, 2020 (1), pp.21-35. ⟨10.1002/ejic.201900810⟩
Journal articles hal-02332497v1
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Atypical McMurry Cross-Coupling Reactions Leading to a New Series of Potent Antiproliferative Compounds Bearing the Key [Ferrocenyl-Ene-Phenol] Motif

Pascal Pigeon , Meral Goermen , Konrad Kowalski , Helge Mueller-Bunz , Michael J. Mcglinchey , et al.
Molecules, 2014, 19 (7), pp.10350-10369. ⟨10.3390/molecules190710350⟩
Journal articles hal-01230372v1
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CDModelTree (V1): Manipulation of a cyclodextrin-ferrociphenol supramolecular models database using a PHP web application

Pascal Pigeon
Software hal-03991394v1
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Enzymatic oxidation of ansa-ferrocifen leads to strong and selective thioredoxin reductase inhibition in vitro

Valeria Scalcon , Anna Citta , Alessandra Folda , Alberto Bindoli , Michèle Salmain , et al.
Journal of Inorganic Biochemistry, 2016, 165, pp.146-151. ⟨10.1016/j.jinorgbio.2016.08.005⟩
Journal articles hal-01401089v1

Imino-tetrahydro-benzothiazole Derivatives as p53 Inhibitors: Discovery of a Highly Potent in Vivo Inhibitor and Its Action Mechanism

Nicolas Pietrancosta , Anice Moumen , Rosanna Dono , Paul Lingor , Veronique Planchamp , et al.
Journal of Medicinal Chemistry, 2006, 49 (12), pp.3645-3652. ⟨10.1021/jm060318n⟩
Journal articles istex hal-02351704v1

Synthesis of New Substituted 4,5-Dihydro-3H-spiro[1,5]-benzoxazepine-2,4′-piperidine and Biological Properties

Younes Laras , Nicolas Pietrancosta , Vincent Moret , Sylvain Marc , Cédrik Garino , et al.
Australian Journal of Chemistry, 2006, 59 (11), pp.812. ⟨10.1071/ch06318⟩
Journal articles hal-02351717v1
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Introducing the Chiral Constrained α‐Trifluoromethylalanine in Aib Foldamers to Control, Quantify and Assign the Helical Screw‐Sense**

Lizeth Bodero , Karine Guitot , Nathalie Lensen , Olivier Lequin , Thierry Brigaud , et al.
Chemistry - A European Journal, 2022, 28 (8), pp.e202103887. ⟨10.1002/chem.202103887⟩
Journal articles hal-03626224v1
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Chemo- and Diastereoselective Hydrosilylation of Amorphadiene toward the Synthesis of Artemisinin

Geoffrey Schwertz , Andrea Zanetti , Marllon Nascimento de Oliveira , Mario Andrés Gomez Fernandez , Zacharias Amara , et al.
Journal of Organic Chemistry, 2020, 85 (15), pp.9607 - 9613. ⟨10.1021/acs.joc.0c00617⟩
Journal articles hal-03290007v1
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A Conjugate between Lqh-8/6, a Natural Peptide Analogue of Chlorotoxin, and Doxorubicin Efficiently Induces Glioma Cell Death

Lucie Dardevet , Feten Najlaoui , Sonia Aroui , Mayeul Collot , Céline Tisseyre , et al.
Biomedicines, 2022, 10 (10), pp.2605. ⟨10.3390/biomedicines10102605⟩
Journal articles hal-03842766v1

Electrochemical primer extension based on polyoxometalate electroactive labels for multiplexed detection of single nucleotide polymorphisms

Nassif Chahin , Laura Uribe , Ahmed Debela , Serge Thorimbert , Bernold Hasenknopf , et al.
Biosensors and Bioelectronics, 2018, 117, pp.201 - 206. ⟨10.1016/j.bios.2018.06.014⟩
Journal articles hal-01878073v1
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Chemoenzymatic synthesis of arabinomannan (AM) glycoconjugates as potential vaccines for tuberculosis

Zhihao Li , Teodora Bavaro , Sara Tengattini , Roberta Bernardini , Maurizio Mattei , et al.
European Journal of Medicinal Chemistry, 2020, 204, pp.112578. ⟨10.1016/j.ejmech.2020.112578⟩
Journal articles hal-02926443v1

Enantioselective Synthesis of Planar Chiral Ferrocifens that Show Chiral Discrimination in Antiproliferative Activity on Breast Cancer Cells

Laura Cunningham , Yong Wang , Chris Nottingham , Jammah Pagsulingan , Gérard Jaouen , et al.
ChemBioChem, 2020, 21 (20), pp.2974-2981. ⟨10.1002/cbic.202000311⟩
Journal articles hal-02771405v1
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Synthesis and Biodistribution of 1-[2-(cyclopentadienyltricarbonyltechnetium-99m)-2- oxo-ethoxy-phenyl]-1,2-di- (p-hydroxyphenyl)but-1-ene for tumor imaging

Tesnim Dallagi , Mouldi Saidi , Gérard Jaouen , Siden Top
Journal of Organometallic Chemistry, 2019, 591, pp.1-6. ⟨10.1016/j.jorganchem.2019.04.006⟩
Journal articles hal-02163476v1

Protective effect of the octadecaneuropeptide on hydrogen peroxide-induced oxidative stress and cell death in cultured rat astrocytes

Yosra Hamdi , Olfa Masmoudi-Kouki , Hadhemi Kaddour , Feten Belhadj , Pierrick Gandolfo , et al.
Journal of Neurochemistry, 2011, 118 (3), pp.416-428. ⟨10.1111/j.1471-4159.2011.07315.x⟩
Journal articles hal-01962753v1

Identification of 26RFa, a hypothalamic neuropeptide of the RFamide peptide family with orexigenic activity

Nicolas Chartrel , Cynthia Dujardin , Youssef Anouar , Jérôme Leprince , Annick Decker , et al.
Proceedings of the National Academy of Sciences of the United States of America, 2011, 100 (25), pp.15247-15252. ⟨10.1073/pnas.2434676100⟩
Journal articles hal-01960798v1

Substituted thiazolamide coupled to a redox delivery system: a new γ-secretase inhibitor with enhanced pharmacokinetic profile

Younes Laras , Gilles Quéléver , Cédrik Garino , Nicolas Pietrancosta , Mahmoud Sheha , et al.
Organic & Biomolecular Chemistry, 2005, 3 (4), pp.612-618. ⟨10.1039/b415090b⟩
Journal articles istex hal-02351730v1

Prospects for the Resistance to HIV Protease Inhibitors: Current Drug Design Approaches and Perspectives

S. Burlet , Nicolas Pietrancosta , Y. Laras , C. Garino , G. Quélever , et al.
Current Pharmaceutical Design, 2005, 11 (24), pp.3077-3090. ⟨10.2174/1381612054864939⟩
Journal articles hal-02351757v1

Novel Tools towards Magnetic Guidance of Neurite Growth: (I) Guidance of Magnetic Nanoparticles into Neurite Extensions of Induced Human Neurons and In Vitro Functionalization with RAS Regulating Proteins

Hendrik Schöneborn , Fabian Raudzus , Emilie Secret , Nils Otten , Aude Michel , et al.
Journal of Functional Biomaterials, 2019, 10 (3), pp.32. ⟨10.3390/jfb10030032⟩
Journal articles hal-02332797v1

The inhibition of tyrosinase by some aryl butenes: A desired activity or a side effect to avoid

Emna E. Ketata , Aref Neifar , Wafa Mihoubi , Pascal Pigeon , Hicham Gouzi , et al.
Journal of Organometallic Chemistry, 2017, 848, pp.133 - 141. ⟨10.1016/j.jorganchem.2017.07.031⟩
Journal articles hal-01611372v1

Efficient ferrocifen anticancer drug and Bcl-2 gene therapy using lipid nanocapsules on human melanoma xenograft in mouse

Pauline Resnier , Natacha Galopin , Yann Sibiril , Anne Clavreul , Jérôme Cayon , et al.
Pharmacological Research, 2017, 126 (19), pp.54 - 65. ⟨10.1016/j.phrs.2017.01.031⟩
Journal articles hal-01878047v1

Synthesis and anti-HIV properties of new hydroxyquinoline–polyamine conjugates on cells infected by HIV-1 LAV and HIV-1 BaL viral strains

Vincent Moret , Nathalie Dereudre-Bosquet , Pascal Clayette , Younes Laras , Nicolas Pietrancosta , et al.
Bioorganic and Medicinal Chemistry Letters, 2006, 16 (23), pp.5988-5992. ⟨10.1016/j.bmcl.2006.08.114⟩
Journal articles istex hal-02351693v1

1,1′-Xylyl bis-1,4,8,11-tetraaza cyclotetradecane: A new potential copper chelator agent for neuroprotection in Alzheimer’s disease. Its comparative effects with clioquinol on rat brain copper distribution

Vincent Moret , Younes Laras , Nicolas Pietrancosta , Cédrik Garino , Gilles Quéléver , et al.
Bioorganic and Medicinal Chemistry Letters, 2006, 16 (12), pp.3298-3301. ⟨10.1016/j.bmcl.2006.03.026⟩
Journal articles istex hal-02351702v1
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Synthèse et étude du mécanisme d’action cytotoxique de complexes organométalliques d’iridium à ligand arène

Robin Ramos
Chimie de coordination. Sorbonne Université, 2021. Français. ⟨NNT : 2021SORUS463⟩
Theses tel-03727628v1
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Heterogeneity of Response to Iron-Based Metallodrugs in Glioblastoma Is Associated with Differences in Chemical Structures and Driven by FAS Expression Dynamics and Transcriptomic Subtypes

Anne Vessieres , Emie Quissac , Nolwenn Lemaire , Agusti Alentorn , Patrycja Domeracka , et al.
International Journal of Molecular Sciences, 2021, 22 (19), pp.10404. ⟨10.3390/ijms221910404⟩
Journal articles hal-03356305v1
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Peptides et Cancers : contribution à l'étude de la carnosine, l'asporine et la thrombospondine

Eva Lardé
Médecine humaine et pathologie. Sorbonne Université; Université de Liège, 2019. Français. ⟨NNT : 2019SORUS520⟩
Theses tel-03400307v1
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Insights into the antiproliferative mechanism of (C^N)-chelated half-sandwich iridium complexes

Robin Ramos , Jeremy Malcolm Zimbron , Serge Thorimbert , Lise-Marie Chamoreau , Annie Munier , et al.
Dalton Transactions, 2020, 49 (48), pp.17635-17641. ⟨10.1039/D0DT03414B⟩
Journal articles hal-03014551v1